2775-2778
De Novo Design of a Novel Oxazolidinone Analogue as a Potent and Selective 
1A Adrenergic Receptor Antagonist with High Oral Bioavailability
2779-2782
3,5-Disubstituted-4-hydroxyphenyls Linked to 3-Hydroxy-2-methyl- 4(1H)-pyridinone: Potent Inhibitors of Lipid Peroxidation and Cell Toxicity
ARTICLES
2783-2788
A Molecular Model for DNA Cross-Linking by the Antitumor Agent Azinomycin B
2789-2796
A Refined 3-Dimensional QSAR of Cytochrome P450 2C9: Computational Predictions of Drug Interactions
2797-2804
Identification of Novel Purine and Pyrimidine Cyclin-Dependent Kinase Inhibitors with Distinct Molecular Interactions and Tumor Cell Growth Inhibition Profiles
2805-2813
Further Studies on Nociceptin-Related Peptides: Discovery of a New Chemical Template with Antagonist Activity on the Nociceptin Receptor
2814-2823
A Novel Class of Highly Potent and Selective A1 Adenosine Antagonists: Structure-Affinity Profile of a Series of 1,8-Naphthyridine Derivatives
2824-2830
Structure-Activity Studies of Reduced-Size Gonadotropin-Releasing Hormone Agonists Derived from the Sequence of an Endothelin Antagonist
2831-2836
Design and Synthesis of Potent Hexapeptide and Heptapeptide Gonadotropin-Releasing Hormone Antagonists by Truncation of a Decapeptide Analogue Sequence
2837-2850
Synthesis of Novel 5-Substituted 3-Amino-3,4-dihydro-2H-1-benzopyran Derivatives and Their Interactions with the 5-HT1A Receptor
2851-2859
Synthesis and Anticonvulsant Activity of Novel and Potent 6,7-Methylenedioxyphthalazin-1(2H)-ones
2860-2870
Ester and Amide Derivatives of the Nonsteroidal Antiinflammatory Drug, Indomethacin, as Selective Cyclooxygenase-2 Inhibitors
2871-2882
Synthesis and Pharmacological Evaluation of Thiopyran Analogues of the Dopamine D3 Receptor-Selective Agonist (4aR,10bR)-(+)-trans-3,4,4a,10b- Tetrahydro-4-n-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol (PD 128907)
2883-2893
Adenosine Kinase Inhibitors. 1. Synthesis, Enzyme Inhibition, and Antiseizure Activity of 5-Iodotubercidin Analogues
2894-2905
Adenosine Kinase Inhibitors. 2. Synthesis, Enzyme Inhibition, and Antiseizure Activity of Diaryltubercidin Analogues
2906-2914
Permanently Charged Chiral 1,4-Dihydropyridines: Molecular Probes of L-Type Calcium Channels. Synthesis and Pharmacological Characterization of Methyl ( 
-Trimethylalkylammonium) 1,4-Dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3,5- pyridinedicarboxylate Iodide, Calcium Channel Antagonists
2915-2921
Synthesis and Biological Evaluation of Certain ,
-Unsaturated Ketones and Their Corresponding Fused Pyridines as Antiviral and Cytotoxic Agents
2922-2928
ElogPoct: A Tool for Lipophilicity Determination in Drug Discovery
2929-2937
Discovery of Novel and Potent Retinoic Acid Receptor Agonists: Syntheses and Evaluation of Benzofuranyl-pyrrole and Benzothiophenyl-pyrrole Derivatives
2938-2945
Synthesis and Evaluation of Peptidomimetics as Selective Inhibitors and Active Site Probes of Nitric Oxide Synthases
2946-2961
Synthesis and Immunosuppressive Activity of 2-Substituted 2-Aminopropane-1,3-diols and 2-Aminoethanols 
BRIEF ARTICLES
2962-2966
Novel Mutual Prodrug of Retinoic and Butyric Acids with Enhanced Anticancer Activity
BOOK REVIEWS
2967-2967
Drugs: Synonyms & Properties Edited by G. W. A. Milne. Ashgate Publishing Co., Burlington, VT. 1999. xx + 1267 pp. 18 x 25.5 cm. ISBN 0-566-8228-4. $250.00.
2967-2968
Biocatalysis Edited by Ramesh N. Patel. Marcel Dekker, New York. 2000. xiii + 932 pp. 17.5 x 25.5 cm. ISBN 0-8247-8282-8. $250.00.
2968-2969
Job$ in the Drug Industry. A Career Guide for Chemists By Richard Friary. Academic Press, San Diego, CA. 2000. xxiii + 364 pp. 15 × 23 cm. ISBN 0-12-267645-9. $39.95.
2969-2969
Metal Ions in Biological Systems. Volume 37. Manganese and Its Role in Biological Processes Edited by Astrid Sigel and Helmut Sigel. Marcel Dekker, New York. 2000. xlvi + 761 pp. 16 × 23.5 cm. ISBN 0-8247-0288-3. $250.00.
2969-2970
The Alkaloids. Volume 52. Chemistry and Biology Edited by Geoffrey A. Cordell. Academic Press, San Diego, CA. 1999. x + 391 pp. 15.5 × 23.5 cm. ISBN 0-12-469552-3. $135.00.